Merck, B2185-10MG, Bisoprolol hemifumarate salt

Name: Bisoprolol hemifumarate salt
Brand: Merck
SKU: B2185-10MG

Size:10 mg, 1-[4-[[2-(1-Methylethoxy)ethoxy]methyl]phenoxy]-3-[(1-methylethyl)amino]-2-propanol hemifumarate salt, ≥98% (HPLC), solid

Available Catalog Numbers

B2185-10MG B2185-50MG

Catalog Number: B2185-10MG

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Category

General Purpose Incubators

Pack Size10 mg

CollectionsMerck Cell Culture Supplements & Reagents: Complete Solutions for Research & Bioproduction Merck Roche Life Science Products for PCR, RT‑PCR & Nucleic Acid Purification

Manufacturer's Pagewww.sigmaaldrich.com/US/en/product/SIGMA/B2185

Description

Application
Bisoprolol hemifumarate salt has been used as a β-adrenergic receptor (β-AR) antagonist in cardiac fibrosis mice model.
Biochem/physiol Actions
Bisoprolol hemifumarate is useful in oral formulations due to its high bioavailability. It also shows long elimination half-life.
Cardioselective β₁-adrenoceptor antagonist.
Features and Benefits
This compound is a featured product for Neuroscience research. Click here to discover more featured Neuroscience products. Learn more about bioactive small molecules for other areas of research at sigma.com/discover-bsm.
This compound was developed by Teva. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.

Specifications

General

UNSPSC Code	12352200
PubChem Substance ID	24724414
NACRES	NA.77
Web Name Suffix Override	≥98% (HPLC), β1-adrenoceptor antagonist, solid
MDL number	MFCD00792743
SMILES string	OC(=O)\C=C\C(O)=O.CC(C)NCC(O)COc1ccc(COCCOC(C)C)cc1.CC(C)NCC(O)COc2ccc(COCCOC(C)C)cc2
InChI key	VMDFASMUILANOL-WXXKFALUSA-N
InChI	1S/2C18H31NO4.C4H4O4/c21-14(2)19-11-17(20)13-23-18-7-5-16(6-8-18)12-21-9-10-22-15(3)4;5-3(6)1-2-4(7)8/h25-8,14-15,17,19-20H,9-13H2,1-4H3;1-2H,(H,5,6)(H,7,8)/b;;2-1+
assay	≥98% (HPLC)
form	solid
color	white
solubility	DMSO: >20 mg/mL
originator	Teva
Gene Information	human ... ADRB1(153)